N-乙基-7,8-二氢-7-甲基-8-氧代-2-苯基-N-(苯基甲基)-9H-嘌呤-9-乙酰胺
Emapunil(AC-5216)
CAS: 226954-04-7
化学式: C23H23N5O2
| 中文名 | Emapunil |
| 英文名 | AC-5216 |
| 别名 | EMAPUNIL游离 EMAPUNIL游离态 N-乙基-7,8-二氢-7-甲基-8-氧代-2-苯基-N-(苯基甲基)-9H-嘌呤-9-乙酰胺 N-苄基-N-乙基-2-(7-甲基-8-氧代-2-苯基-7,8-二氢-9H-嘌呤-9-基)乙酰胺 |
| 英文别名 | XBD-173 AC-5216 Emapunil EMapunil Emapunil(AC-5216) AC 5216 (Emapunil) N-Benzyl-N-ethyl-2-(7-Methyl-8-oxo-2-phenyl-7,8-dihydro-9H-purin-9-yl)acetaMide N-Ethyl-7,8-dihydro-7-methyl-8-oxo-2-phenyl-N-(phenylmethyl)-9H-purine-9-acetamide 9H-Purine-9-acetaMide,N-ethyl-7,8-dihydro-7-Methyl-8-oxo-2-phenyl-N-(phenylMethyl)- |
| CAS | 226954-04-7 |
| 化学式 | C23H23N5O2 |
| 分子量 | 401.46 |
| 存储条件 | 2-8°C |
| 外观 | 粉末 |
| 颜色 | white to beige |
| 体内研究 | Emapunil (AC-5216, 0.1-3, 0.003-0.01 and 0.01-0.3 mg/kg, p.o.) produces anti-anxiety effects in the Vogel-type conflict test in rats, and in the light/dark box and social interaction tests in mice. Emapunil (AC-5216, 3-30 mg/kg, p.o.) reduces the immobility time, and this effect was blocked by PK11195. Emapunil (AC-5216, 1-100 mg/kg, p.o.) produces no distinct change in the rat electroencephalogram. Emapunil (AC-5216, 0.3 and 1 mg/kg, i.g.) causes significant suppression of the enhanced anxiety and contextual fear induced in post-TDS rats. Emapunil (AC-5216, 0.3 and 1 mg/kg, i.g.) alleviates the enhanced anxiety and fear response in a time-dependent sensitization (TDS) procedure, a rat PTSD animal model. Emapunil (AC-5216, 0.3 and 1 mg/kg, i.g.) reverses the increased plasma glucose (PG) and decreased insulin (INS) in HFD-STZ rats. Animal Model: Rats. Dosage: 0.1-3 mg/kg. Administration: P.O.. Result: Significantly increased the number of shocks that rats received. Significantly increased the time spent in the light compartment but only slightly increased that time at 0.03 mg/kg, p.o. (P<0.1). |
N-乙基-7,8-二氢-7-甲基-8-氧代-2-苯基-N-(苯基甲基)-9H-嘌呤-9-乙酰胺 - 配置溶液浓度参考
| 1mg | 5mg | 10mg | |
|---|---|---|---|
| 1 mM | 2.491 ml | 12.454 ml | 24.909 ml |
| 5 mM | 0.498 ml | 2.491 ml | 4.982 ml |
| 10 mM | 0.249 ml | 1.245 ml | 2.491 ml |
| 5 mM | 0.05 ml | 0.249 ml | 0.498 ml |
最后更新：2024-01-02 23:10:35
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现货供应
产品名: N-苄基-N-乙基-2-(7-甲基-8-氧代-2-苯基-7,8-二氢-9H-嘌呤-9-基)乙酰胺 去供应商网站查看 询盘CAS: 226954-04-7
产地: 北京
包装: 瓶
规格: YS152730-5mg,YS152730-10mg
价格: 电话、微信、QQ、邮件
库存: 一周左右
电话: 010-50973130
手机: 17801761073(微信同号)
电子邮件: 3193328036@qq.com
QQ: 3193328036
微信: 17801761073
产品描述: 索莱宝直销，欢迎来询
现货供应
产品名: Emapunil游离态 去供应商网站查看 询盘CAS: 226954-04-7
产地: 中国上海
包装: 10mg
规格: 98%
价格: 1337.00
库存: 10个工作日
电话: 400-900-4166
手机: 18017137653
电子邮件: 3007523013@qq.com
QQ: 3007523013
微信: 18017137653
产品描述: 中文名：Emapunil游离态 英文名:AC-5216 CAS:226954-04-7 规格:98% 产地:中国上海
现货供应
产品名: N-苄基-N-乙基-2-(7-甲基-8-氧代-2-苯基-7,8-二氢-9H-嘌呤-9-基)乙酰胺 去供应商网站查看 询盘CAS: 226954-04-7
产地: 北京
包装: 瓶
规格: YS152730-5mg,YS152730-10mg
价格: 电话、微信、QQ、邮件
库存: 一周左右
电话: 010-50973130
手机: 17801761073(微信同号)
电子邮件: 3193328036@qq.com
QQ: 3193328036
微信: 17801761073
产品描述: 索莱宝直销，欢迎来询
现货供应
产品名: Emapunil游离态 去供应商网站查看 询盘CAS: 226954-04-7
产地: 中国上海
包装: 10mg
规格: 98%
价格: 1337.00
库存: 10个工作日
电话: 400-900-4166
手机: 18017137653
电子邮件: 3007523013@qq.com
QQ: 3007523013
微信: 18017137653
产品描述: 中文名：Emapunil游离态 英文名:AC-5216 CAS:226954-04-7 规格:98% 产地:中国上海
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