中文名 | NETAMIFTIDE |
英文名 | NETAMIFTIDE |
英文别名 | NETAMIFTIDE Nemifitide di INN 00835 diTFA Nemifitide diTFA NEMIFITIDE DITFA Bis(trifluoroacetate) Netamiftide ditriflutate FLUORO-PHE-HYP-ARG-GLY-TRP-NH2 (2S)-N-[(1S)-1-[[(1S)-1-[[(2S)-2-amino-3-(4-fluorophenyl)propanoyl]carbamoyl]-2-(1H-indol-3-yl)ethyl]carbamoylmethylcarbamoyl]-4-(diaminomethylideneamino)butyl]-4-hydroxy-pyrrolidine-2-carboxamide |
CAS | 204992-09-6 |
化学式 | C37H45F7N10O10 |
体外研究 | Nemifitide diTFA (INN 00835 diTFA) and its active metabolite (M1) bind at micromolar concentrations to several receptors including the 5-HT 2A , 5-HT 2C , melanocortin MC4, MC5 and bombesin. |
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