GRK2 inhibitor GS180736A
GSK180736A
CAS: 817194-38-0
Molecular Formula: C19H16FN5O2
GRK2 inhibitor GS180736A - Names and Identifiers
GRK2 inhibitor GS180736A - Physico-chemical Properties
| Molecular Formula | C19H16FN5O2 |
| Molar Mass | 365.36 |
| Solubility | DMSO: ≥ 30 mg/mL |
| Storage Condition | -20℃ |
| In vitro study | GSK180736A inhibited GRK2 with an IC50 of 770 nM, 300 times more potent than grk5. It is a weak PKA inhibitor with IC50 = 30 μm; However, it is a potent ROCK1 inhibitor (IC50=100 nM). |
GRK2 inhibitor GS180736A - Preparation solution concentration reference
| 1mg | 5mg | 10mg | |
|---|---|---|---|
| 1 mM | 2.737 ml | 13.685 ml | 27.37 ml |
| 5 mM | 0.547 ml | 2.737 ml | 5.474 ml |
| 10 mM | 0.274 ml | 1.369 ml | 2.737 ml |
| 5 mM | 0.055 ml | 0.274 ml | 0.547 ml |
Last Update：2024-01-02 23:10:35
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CAS: 817194-38-0
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CAS: 817194-38-0
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Mobile: 18021002903
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