| Molecular Formula | C27H26N4O2S |
| Molar Mass | 470.59 |
| Storage Condition | Sealed in dry,2-8°C |
| 1mg | 5mg | 10mg | |
|---|---|---|---|
| 1 mM | 2.125 ml | 10.625 ml | 21.25 ml |
| 5 mM | 0.425 ml | 2.125 ml | 4.25 ml |
| 10 mM | 0.213 ml | 1.063 ml | 2.125 ml |
| 5 mM | 0.043 ml | 0.213 ml | 0.425 ml |
| biological activity | TCS 1102 is an orexin OX receptor antagonist, and Ki for OX2 and OX1 receptors are 0.2 and 3 nM respectively. |