| Molecular Formula | C22H29ClN4O3 |
| Molar Mass | 432.94 |
| Density | 1.357±0.06 g/cm3(Predicted) |
| Boling Point | 691.6±55.0 °C(Predicted) |
| Solubility | DMSO: ≥ 71 mg/mL |
| pKa | 9.47±0.50(Predicted) |
| Storage Condition | -20℃ |
| In vitro study | Positive for KRAS mutation (KRAS). ARS853 in the expression of KRAS. |
| 1mg | 5mg | 10mg | |
|---|---|---|---|
| 1 mM | 2.31 ml | 11.549 ml | 23.098 ml |
| 5 mM | 0.462 ml | 2.31 ml | 4.62 ml |
| 10 mM | 0.231 ml | 1.155 ml | 2.31 ml |
| 5 mM | 0.046 ml | 0.231 ml | 0.462 ml |