中文名 | Evifacotrep |
英文名 | 4-chloro-5-{4-[4-fluoro-2-(trifluoromethyl)phenoxy]-5,8-dihydropyrido[3,4-d]pyrimidin-7(6H)-yl}pyridazin-3(2H)-one |
别名 | 依法曲普 |
英文别名 | Evifacotrep 5-chloro-4-[4-[4-fluoro-2-(trifluoromethyl)phenoxy]-6,8-dihydro-5H-pyrido[3,4-d]pyrimidin-7-yl]-1H-pyridazin-6-one 4-chloro-5-{4-[4-fluoro-2-(trifluoromethyl)phenoxy]-5,8-dihydropyrido[3,4-d]pyrimidin-7(6H)-yl}pyridazin-3(2H)-one 3(2H)-Pyridazinone, 4-chloro-5-[4-[4-fluoro-2-(trifluoromethyl)phenoxy]-5,8-dihydropyrido[3,4-d]pyrimidin-7(6H)-yl]- |
CAS | 2413739-88-3 |
化学式 | C18H12ClF4N5O2 |
分子量 | 441.77 |
存储条件 | -20℃ |
产品用途 | vifacotrep is a short transient receptor potential channel 5 (TRPC5) antagonist. |
靶点 | TRPC5 |
1mg | 5mg | 10mg | |
---|---|---|---|
1 mM | 2.264 ml | 11.318 ml | 22.636 ml |
5 mM | 0.453 ml | 2.264 ml | 4.527 ml |
10 mM | 0.226 ml | 1.132 ml | 2.264 ml |
5 mM | 0.045 ml | 0.226 ml | 0.453 ml |
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