Molecular Formula | C44H69N15O9S |
Molar Mass | 984.18 |
Density | 1.42±0.1 g/cm3(Predicted) |
pKa | 9.97±0.15(Predicted) |
Storage Condition | −20°C |
In vitro study | Adrenorphin (Metorphamide) is a opioid octapeptide from bovine brain, acts as a potent agonist of μ-opioid receptor, with K i of 12 nM. The binding ratios of K i for μ-opioid receptor/K i for δ-opioid receptor of 0.04 and of K i for μ-opioid receptor/K i for κ-opioid receptor of 0.46. Adrenorphin potently inhibits catecholamine secretion evoked by 10 μM nicotine in cultured human pheochromocytoma 6 cells, with an IC 50 of 1.1 μM. |
WGK Germany | 3 |