Name | BET-IN-4 |
Synonyms | ODM-207 BET-IN-4 2(1H)-Quinolinone, 6-(3,5-dimethyl-4-isoxazolyl)-7-methoxy-3-methyl-1-(2-pyridinylmethyl)- |
CAS | 1801503-93-4 |
Molecular Formula | C22H21N3O3 |
Molar Mass | 375.42 |
Density | 1.232±0.06 g/cm3(Predicted) |
Boling Point | 529.0±50.0 °C(Predicted) |
pKa | 4.36±0.12(Predicted) |
introduction | ODM-207 is a highly effective, selective and orally active pan-BET inhibitor, which has shown preclinical evidence of tumor growth inhibition in breast cancer, leukemia and prostate cancer xenograft models. |