CS-1645
SR9243
CAS: 1613028-81-1
Molecular Formula: C31H32BrNO4S2
CS-1645 - Names and Identifiers
| Name | SR9243 |
| Synonyms | SR9243 CS-1645 SR 9243 SR-9243 N-(3-bromophenethyl)-2,4,6-trimethyl-N-((3'-(methylsulfonyl)-[1,1'-biphenyl]-4-yl)methyl)benzenesulfonamide N-[2-(3-Bromophenyl)ethyl]-2,4,6-trimethyl-N-[[3'-(methylsulfonyl)[1,1'-biphenyl]-4-yl]methyl]benzenesulfonamide Benzenesulfonamide, N-[2-(3-bromophenyl)ethyl]-2,4,6-trimethyl-N-[[3'-(methylsulfonyl)[1,1'-biphenyl]-4-yl]methyl]- |
| CAS | 1613028-81-1 |
CS-1645 - Physico-chemical Properties
| Molecular Formula | C31H32BrNO4S2 |
| Molar Mass | 626.62 |
| Density | 1.347±0.06 g/cm3(Predicted) |
| Melting Point | 154-155°C |
| Boling Point | 786.3±70.0 °C(Predicted) |
| Solubility | 10 mM in DMSO |
| Appearance | solid |
| Color | White |
| pKa | -6.90±0.70(Predicted) |
| Storage Condition | 2-8°C |
| Stability | Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20° for up to 3 months. |
| In vitro study | In HEK293 cells expressing LXRs, SR9243 inhibits LXR activation by enhancing LXR-co-repressor aggregation. In various cancer cell types, SR9243 reduces cancer cell activity, induces apoptotic cell death, and sensitizes cancer cells to chemotherapy. |
| In vivo study | SR9243 (60 mg/kg, I. p.) inhibits LXR-dependent fat synthase gene expression and tumor growth in Ob/Ob mice fed a high-fat diet. |
CS-1645 - Risk and Safety
| HS Code | 29350090 |
CS-1645 - Preparation solution concentration reference
| 1mg | 5mg | 10mg | |
|---|---|---|---|
| 1 mM | 1.596 ml | 7.979 ml | 15.959 ml |
| 5 mM | 0.319 ml | 1.596 ml | 3.192 ml |
| 10 mM | 0.16 ml | 0.798 ml | 1.596 ml |
| 5 mM | 0.032 ml | 0.16 ml | 0.319 ml |
Last Update：2024-01-02 23:10:35
CS-1645 - Reference Information
| biological activity | SR9243 is a potent and selective inverse agonist of LXR. |
| Target | Value |
Last Update：2024-04-09 21:54:55
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Spot supply
Product Name: SR9243 Visit Supplier Webpage Request for quotationCAS: 1613028-81-1
Tel: 18301782025
Email: 3008007409@qq.com
Mobile: 18021002903
QQ: 3008007409
Wechat: 18301782025
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