Name | MSX-122 |
Synonyms | MSX122 CS-2430 MSX 222 MSX 122 MSX-122 1,4-Benzenedimethanamine, N1,N4-di-2-pyrimidinyl- N-[[4-[(pyrimidin-2-ylamino)methyl]phenyl]methyl]pyrimidin-2-amine |
CAS | 897657-95-3 |
Molecular Formula | C16H16N6 |
Molar Mass | 292.35 |
Density | 1.313±0.06 g/cm3(Predicted) |
Melting Point | 219 °C |
Boling Point | 566.9±60.0 °C(Predicted) |
Solubility | 10 mM in DMSO |
pKa | 3.82±0.10(Predicted) |
Storage Condition | -20℃ |
1mg | 5mg | 10mg | |
---|---|---|---|
1 mM | 3.421 ml | 17.103 ml | 34.207 ml |
5 mM | 0.684 ml | 3.421 ml | 6.841 ml |
10 mM | 0.342 ml | 1.71 ml | 3.421 ml |
5 mM | 0.068 ml | 0.342 ml | 0.684 ml |
biological activity | MSX-122 is a new type of CXCR4 partial antagonist with an IC50 of about 10 nM. |
target | TargetValue CXCR4 () ~ 10 nM |
Target | Value |
CXCR4 () | ~10 nM |