PF-04981517
PF-4981517
CAS: 1390637-82-7
Molecular Formula: C26H32N8
PF-04981517 - Names and Identifiers
PF-04981517 - Physico-chemical Properties
| Molecular Formula | C26H32N8 |
| Molar Mass | 456.59 |
| Appearance | powder |
| Color | white to beige |
| Storage Condition | room temp |
| In vitro study | PF-4981517 (cyp3ide) is a highly potent, time-specific inhibitor of human CYP3A4. PF-4981517 reversible inhibition of some human cytochrome P450 activities. PF-4981517 acts on CYP3A4, 3A5, and 3A7 with an IC50 of 0.03 μm, 17 μm, and 70 μm, respectively. PF-4981517 co-inhibited all CYP3A activity with Ketoconazole. |
PF-04981517 - Risk and Safety
| WGK Germany | 3 |
PF-04981517 - Reference Information
| biological activity | PF-4981517 (CYP3cide, PF-04981517) is an effective and selective CYP3A4(P450) inhibitor with an IC50 of 0.03 μM, which is more than 500 times more selective than CYP3A5 and CYP3A7. |
| target | TargetValue CYP3A4 30 nM |
| Target | Value |
| CYP3A4 | 30 nM |
| In vitro studies | PF-4981517(CYP3cide) is a highly effective, time-dependent human CYP3A4 inhibitor. PF-4981517 reversibly inhibits some human cytochrome P450 activities. PF-4981517 act on CYP3A4, 3A5, and 3A7, IC50 are 0.03 μM, 17 μM, and 70 μM, respectively. PF-4981517 and Ketoconazole together inhibit all CYP3A activities. |
Last Update：2024-04-09 21:54:55
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CAS: 1390637-82-7
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Product Name: PF-4981517 Visit Supplier Webpage Request for quotation
CAS: 1390637-82-7
Tel: 18301782025
Email: 3008007409@qq.com
Mobile: 18021002903
QQ: 3008007409
Wechat: 18301782025
CAS: 1390637-82-7
Tel: 18301782025
Email: 3008007409@qq.com
Mobile: 18021002903
QQ: 3008007409
Wechat: 18301782025
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