Name | SIRAMESINE |
Synonyms | CS-1476 SIRAMESINE 1'-[4-[1-(4-fluorophenyl)indol-3-yl]butyl]spiro[1H-2-benzofuran-3,4'-piperidine] 1'-(4-(1-(4-fluorophenyl)-1H-indol-3-yl)butyl)-3H-spiro[isobenzofuran-1,4'-piperidine] Spiro[isobenzofuran-1(3H),4'-piperidine], 1'-[4-[1-(4-fluorophenyl)-1H-indol-3-yl]butyl]- 1'-[4-[1-(4-Fluorophenyl)-1H-indol-3-yl]-1-butyl]spiro[isobenzofuran-1(3H),4'-piperidine] 1'-(4-(1-(4-FLUOROPHENYL)-1H-INDOL-3-YL)BUTYL)-3H-SPIRO[ISOBENZOFURAN-1,4'-PIPERIDINE].HCL |
CAS | 147817-50-3 |
Molecular Formula | C30H31FN2O |
Molar Mass | 454.58 |
Density | 1.19±0.1 g/cm3(Predicted) |
Boling Point | 611.4±55.0 °C(Predicted) |
Solubility | Soluble in DMSO (up to at least 25 mg/ml) |
Appearance | solid |
Color | White |
pKa | 9.45±0.20(Predicted) |
Storage Condition | Sealed in dry,Room Temperature |
Stability | Stable for 1 year from date of purchase as supplied. Solutions in DMSO may be stored at -20°C for up to 3 months. |
1mg | 5mg | 10mg | |
---|---|---|---|
1 mM | 2.2 ml | 10.999 ml | 21.998 ml |
5 mM | 0.44 ml | 2.2 ml | 4.4 ml |
10 mM | 0.22 ml | 1.1 ml | 2.2 ml |
5 mM | 0.044 ml | 0.22 ml | 0.44 ml |
Biological activity | Siramesine(Lu 28-179) is a sigma-2 receptor agonist that can cause the death of cancer cells and has anti-cancer activity in the body. |