LKB1/AAK1 dual inhibitor MedChemExpress (MCE)

Product Name	Pim1/AKK1-IN-1
Synonyms	CS-2864 3-B]PYRIDIN-3-YL]- 3-b]pyridin-3-yl]- AAK1 DUAL INHIBITOR 3-PYRIDINECARBOXAMIDE LKB1(AAK1 dual inhibitor) N-[5-(4-cyanophenyl)-1H-pyrrolo[2 Synonyms CS-2864 3-B]PYRIDIN-3-YL]- 3-b]pyridin-3-yl]- AAK1 DUAL INHIBITOR 3-PYRIDINECARBOXAMIDE LKB1(AAK1 dual inhibitor) N-[5-(4-cyanophenyl)-1H-pyrrolo[2 N-[5-(4-CYANOPHENYL)-1H-PYRROLO[2 N-[5-(4-Cyanophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]-3-pyridinecarboxamide
CAS	1093222-27-5
EINECS
Chemical Formula	C20H13N5O
Molecular Weight	339.35
inchi
Package	10 mM * 1 mL;1 mg;5 mg;10 mg;25 mg;50 mg
Price	Email to quote
Descriptions	Pim1/AKK1-IN-1 Pim1/AKK1-IN-1 MedChemExpress (MCE) HY-10371 1093222-27-5 LKB1/AAK1 dual inhibitor 98.40% Powder -20°C 3 years 4°C 2 years In solvent -80°C 2 years -20°C 1 year Room temperature in continental US Descriptions Pim1/AKK1-IN-1 Pim1/AKK1-IN-1 MedChemExpress (MCE) HY-10371 1093222-27-5 LKB1/AAK1 dual inhibitor 98.40% Powder -20°C 3 years 4°C 2 years In solvent -80°C 2 years -20°C 1 year Room temperature in continental US may vary elsewhere. Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and also inhibits MPSK1 and TNIK. Pim1/AKK1-IN-1 is multi-kinase inhibitor, and has Kd of 380 nM against LKB1 and 53 nM against AAK1[1]. PIM1 \| \| \| \| \| \| \| \| \| \| [1]. Bamborough P, et al. Assessment of chemical coverage of kinome space and its implications for kinase drug discovery. J Med Chem. 2008 Dec 25 51(24):7898-914. [Content Brief]
Last Update	2025-04-01 14:45:47

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