Org-8282 MedChemExpress (MCE)

Product Name	Setiptiline
Synonyms	Tecipul;Org-8282;Setiptiline;Teciptiline;Teciptilline;Setiptiline(Teciptilline)
CAS	57262-94-9
EINECS	260-653-4
Chemical Formula	C19H19N
Molecular Weight	261.36
inchi
Package	10 mM * 1 mL;50 mg;100 mg
Price	Email to quote
Descriptions	Setiptiline Setiptiline MedChemExpress (MCE) HY-32329 57262-94-9 Org-8282 98.03% Powder -20°C 3 years 4°C 2 years In solvent -80°C 2 years -20°C 1 year Room temperature in continental US Descriptions Setiptiline Setiptiline MedChemExpress (MCE) HY-32329 57262-94-9 Org-8282 98.03% Powder -20°C 3 years 4°C 2 years In solvent -80°C 2 years -20°C 1 year Room temperature in continental US may vary elsewhere. Setiptiline (Org-8282) is a serotonin receptor antagonist. Setiptiline is a tetracyclic antidepressant (TeCA) which acts as a noradrenergic and specific serotonergic antidepressant (NaSSA). Setiptiline acts as a norepinephrine reuptake inhibitor, α2-adrenergic receptor antagonist, and serotonin receptor antagonist, likely at the 5-HT2A, 5-HT2C, and/or 5-HT3 subtypes, as well as an H1 receptor inverse agonist/antihistamine. 5-HT2A Receptor 5-HT2C Receptor 5-HT3 Receptor \| \| \| \| \| \| \| \| \| \| [1]. Yamada K, Furukawa T. [Behavioral effects of a new antidepressant, setiptiline]. Nihon Yakurigaku Zasshi. 1991 Jan 97(1):31-9. [Content Brief] [2]. Kamimura M, Aoba A, Yamaguchi N et al. The effect of age on plasma level of setiptiline maleate in depressed patients. Prog Neuropsychopharmacol Biol Psychiatry. 1994 Oct 18(6):1015-26. [Content Brief] [3]. Kuniyoshi M, Nakamura J, Miura C, Inanaga K. Effectiveness of concomitant setiptiline maleate (Tecipul) on negative symptoms of schizophrenia. Prog Neuropsychopharmacol Biol Psychiatry. 1994 Mar 18(2):339-46. [Content Brief] [4]. Niho T, Ito C, Shibutani Y, Hashizume H, Yamaguchi K. [Pharmacological properties of MO-8282, a novel antidepressant]. Nihon Yakurigaku Zasshi. 1986 Oct 88(4):309-20. [Content Brief]
Last Update	2025-04-01 14:45:47

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