Y-25130 hydrochloride MedChemExpress (MCE)

Product Name	Azasetron hydrochloride
Synonyms	Y-25130 Azasetron HCl AZASETRON HCL Azasetron base Y-25130 HYDROCHLORIDE Azasetron hydrochloride n-(1-azabicyclo[2.2.2]octan-8-yl)-6-chloro-4-methyl-3-oxo-1,4-benzoxazine-8-carboxamide hydrochloride Synonyms Y-25130 Azasetron HCl AZASETRON HCL Azasetron base Y-25130 HYDROCHLORIDE Azasetron hydrochloride n-(1-azabicyclo[2.2.2]octan-8-yl)-6-chloro-4-methyl-3-oxo-1,4-benzoxazine-8-carboxamide hydrochloride N-(1-AZABICYCLO[2.2.2]OCT-3-YL)-6-CHLORO-4-METHYL-3-OXO-3,4-DIHYDRO-2H-1,4-BENZOXAZINE-8-CARBOXAMIDE HCL n-1-azabicyclo[2.2.2]oct-3-yl-6-chloro-3,4-dihydro-4-methyl-3-oxo-2h-1,4-benzoxazine-8-carboxamide hydrochloride N-(1-azabicyclo[2.2.2]oct-3-yl)-6-chloro-4-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazine-8-carboxamide hydrochloride N-(1-AZABICYCLO[2.2.2]OCT-3-YL)-6-CHLORO-4-METHYL-3-OXO-3,4-DIHYDRO-2H-1,4-BENZOXAZINE-8-CARBOXAMIDE hydrochloride N-(1-AZABICYCLO[2.2.2]OCT-3-YL)-6-CHLORO-4-METHYL-3-OXO-3,4-DIHYDRO-2H-1,4-BENZOXAZINE-8-CARBOXAMIDE HYDROCHLORIDE N-1-AZABICYCLO[2.2.2]-OCT-3-YL-6-CHLORO-3,4-DIHYDRO-4-METHYL-3-OXO-2H-1,4-BENZOXAZINE-8-CARBOXAMIDE, HYDROCHLORIDE
CAS	123040-69-7;123040-16-4;141922-90-9
EINECS	1533716-785-6
Chemical Formula	C17H20ClN3O3
Molecular Weight	349.81
inchi	InChI=1/C17H20ClN3O3.ClH/c1-20-14-7-11(18)6-12(16(14)24-9-15(20)22)17(23)19-13-8-21-4-2-10(13)3-5-21;/h6-7,10,13H,2-5,8-9H2,1H3,(H,19,23);1H
Package	10 mM * 1 mL;5 mg;10 mg;50 mg;100 mg
Price	Email to quote
Descriptions	Azasetron hydrochloride Azasetron hydrochloride MedChemExpress (MCE) HY-B0068 123040-16-4 Y-25130 hydrochloride 99.76% 4°C, sealed storage, away from moisture In solvent : -80°C, 6 months Descriptions Azasetron hydrochloride Azasetron hydrochloride MedChemExpress (MCE) HY-B0068 123040-16-4 Y-25130 hydrochloride 99.76% 4°C, sealed storage, away from moisture In solvent : -80°C, 6 months -20°C, 1 month (sealed storage, away from moisture) Room temperature in continental US may vary elsewhere. Azasetron (Y-25130) hydrochloride, a benzamide derivative, is a potent and selective 5-HT3 receptor antagonist. Azasetron is used in the study for Chemotherapy-induced nausea and vomiting (CINV). Azasetron could effectively penetrate through the skin and pass into the systemic circulation[2]. 5-HT3 Receptor 0.33 nM (IC50) \| \| \| \| \| \| \| \| \| \| [1]. Sato, N., et al., Antagonistic activity of Y-25130 on 5-HT3 receptors. Jpn J Pharmacol, 1992. 59(4): p. 443-8. [Content Brief] [2]. Haga, K., et al., The effects of orally administered Y-25130, a selective serotonin3-receptor antagonist, on chemotherapeutic agent-induced emesis. Jpn J Pharmacol, 1993. 63(3): p. 377-83. [Content Brief]
Last Update	2025-04-01 14:45:47

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