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Supplier NameMedChemExpress (MCE)
Contactsales
Tel609-228-6898
Mobile609-228-6898
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Emailsales@medchemexpress.com; tech@medchemexpress.com
Websitehttps://www.medchemexpress.com/
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Product NameGSK6853
SynonymsGSK6853
CS-2243
GSK-6853
GSK 6853
FQWDVNSBYDXPIO-CQSZACIVSA-N
BRPF1 bromodomain inhibitor GS6853
N-[2,3-dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide

Synonyms

GSK6853
CS-2243
GSK-6853
GSK 6853
FQWDVNSBYDXPIO-CQSZACIVSA-N
BRPF1 bromodomain inhibitor GS6853
N-[2,3-dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxybenzamide
Benzamide, N-[2,3-dihydro-1,3-dimethyl-6-[(2R)-2-methyl-1-piperazinyl]-2-oxo-1H-benzimidazol-5-yl]-2-methoxy-
CAS1910124-24-1
EINECS
Chemical FormulaC22H27N5O3
Molecular Weight409.48
inchi
Package10 mM * 1 mL;1 mg;5 mg;10 mg;25 mg;50 mg;100 mg
PriceEmail to quote
DescriptionsGSK6853

GSK6853

MedChemExpress (MCE)

HY-100220

1910124-24-1

99.89%

Powder -20°C 3 years 4°C 2 years In solvent -80°C 2 years -20°C 1 year

Room temperature in continental US

Descriptions

GSK6853

GSK6853

MedChemExpress (MCE)

HY-100220

1910124-24-1

99.89%

Powder -20°C 3 years 4°C 2 years In solvent -80°C 2 years -20°C 1 year

Room temperature in continental US
may vary elsewhere.

GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain.

The ip route of administration would be suitable for dosing GSK6853 in potential PK/PD models[1].

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[1]. Bamborough P et al. GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain. ACS Med Chem Lett. 2016 May 9
7(6):552-7. [Content Brief]

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